SCHEMBL8668643

SCHEMBL8668643

CC(=O)Nc1cc2c(cc1Br)CC(NC(C)=O)C2

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.50
CA2 P00918 5/20 0.50
CA12 O43570 3/20 0.50
CA7 P43166 3/20 0.50
CA14 Q9ULX7 3/20 0.50
CA9 Q16790 3/20 0.50
MTNR1A P48039 7/20 0.42
MTNR1B P49286 5/20 0.42
RXFP1 Q9HBX9 1/20 0.37
APOB P04114 1/20 0.37
MTTP P55157 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11985027 0.84 CA1 (0.43) CA1CA2CA12CA7CA14
SCHEMBL8699267 0.78 CA1 (0.38) CA1CA2CA9RXFP1
SCHEMBL19995817 0.77 CA1 (0.45) CA1CA2CA9RXFP1
SCHEMBL29575116 0.77 CA1 (0.45) CA1CA2CA9RXFP1
SCHEMBL433839 0.77 CA1 (0.45) CA1CA2CA9RXFP1
SCHEMBL8667950 0.77 CA1 (0.38) CA1CA2CA9RXFP1
SCHEMBL9093950 0.76 CA1 (0.37) CA1CA2CA12CA7CA14
SCHEMBL18750435 0.75 CA1 (0.56) CA1CA2CA9RXFP1
SCHEMBL8699261 0.75 CA1 (0.47) CA1CA2CA12CA7CA14
SCHEMBL4808483 0.74 CA1 (0.61) CA1CA2CA12CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO claimed
US-5721234-A TREATING CONVULSIONS, ANXIETY, CEREBRAL HYPOXIA/ISCHEMIA, PARKINSON*S DISEASE WARNER-LAMBERT COMPANY (US) 1998-02-24 US disclosed
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed