SCHEMBL8699267

SCHEMBL8699267

CC(=O)Nc1cc2c(cc1Br)CC(N(C)C(C)=O)C2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
NPY5R Q15761 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAOA P21397 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.31
MAPT P10636 2/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
IDO1 P14902 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11985027 0.80 CA1 (0.43) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL8668643 0.78 CA1 (0.50) CA1CA2CA9RXFP1
SCHEMBL8703459 0.75 NPY5R (0.48) CA1CA2CA9NPY5RALDH1A1
SCHEMBL8133151 0.75 FYN (0.57) MEN1KMT2AMAPT
SCHEMBL19995817 0.73 CA1 (0.45) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL433839 0.73 CA1 (0.45) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL29575116 0.73 CA1 (0.45) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL8667950 0.73 CA1 (0.38) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL18750435 0.72 CA1 (0.56) CA1CA2CA9RXFP1ALDH1A1
SCHEMBL16769416 0.70 CA1 (0.45) CA1CA2CA9RXFP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed