SCHEMBL8669254

SCHEMBL8669254

Nc1c(Br)cc2c(c1[N+](=O)[O-])CC(C(=O)O)C2

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
CTSB P07858 1/20 0.33
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8669853 0.80 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSB
SCHEMBL8669857 0.80 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSB
SCHEMBL8671076 0.80 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSB
Hydrochloric Acid SCHEMBL8668055 0.79 ALDH1A1 (0.38) ALDH1A1CYP3A4CTSB
SCHEMBL8702721 0.79 ALDH1A1 (0.32) ALDH1A1CYP3A4
SCHEMBL8702726 0.79 ALDH1A1 (0.32) ALDH1A1CYP3A4
SCHEMBL8668636 0.77 CA1 (0.44) ALDH1A1CYP3A4
SCHEMBL8675657 0.74 FYN (0.37) ALDH1A1CYP3A4CTSBLMNACYP1A2
SCHEMBL8668680 0.73 FYN (0.39) ALDH1A1CYP3A4CTSBLMNACYP1A2
SCHEMBL21962340 0.71 GRIN1 (0.48) ALDH1A1CYP3A4CTSBTDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721234-A TREATING CONVULSIONS, ANXIETY, CEREBRAL HYPOXIA/ISCHEMIA, PARKINSON*S DISEASE WARNER-LAMBERT COMPANY (US) 1998-02-24 US disclosed
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed