SCHEMBL8669853

SCHEMBL8669853

Nc1c(Br)cc2c(c1[N+](=O)[O-])C[C@H](N)C2

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
CTSB P07858 1/20 0.36
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
CA12 O43570 2/20 0.34
CA7 P43166 2/20 0.34
CA14 Q9ULX7 2/20 0.34
MAPT P10636 1/20 0.31
FYN P06241 1/20 0.31
KCNH2 Q12809 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8669857 1.00 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSBCA1CA2
SCHEMBL8671076 1.00 ALDH1A1 (0.39) ALDH1A1CYP3A4CTSBCA1CA2
Hydrochloric Acid SCHEMBL8668055 0.98 ALDH1A1 (0.38) ALDH1A1CYP3A4CTSBCA1CA2
SCHEMBL8669254 0.80 THRA (0.38) ALDH1A1CYP3A4CTSB
Hydrochloric Acid SCHEMBL8704912 0.79 CA1 (0.33) ALDH1A1CA1CA2CA12CA7
SCHEMBL8675657 0.78 FYN (0.37) ALDH1A1CYP3A4CTSBMAPTFYN
SCHEMBL8668680 0.77 FYN (0.39) ALDH1A1CYP3A4CTSBMAPTFYN
SCHEMBL8668636 0.76 CA1 (0.44) ALDH1A1CYP3A4CA1CA2CA12
SCHEMBL8702726 0.75 ALDH1A1 (0.32) ALDH1A1CYP3A4
SCHEMBL8702721 0.75 ALDH1A1 (0.32) ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721234-A TREATING CONVULSIONS, ANXIETY, CEREBRAL HYPOXIA/ISCHEMIA, PARKINSON*S DISEASE WARNER-LAMBERT COMPANY (US) 1998-02-24 US disclosed
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed