SCHEMBL8669505

SCHEMBL8669505

Cc1cn2cccc(OC(NC(=O)CNC(=O)N(C)c3ccccc3)c3c(Cl)cccc3Cl)c2n1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.33
BDKRB2 P30411 6/20 0.32
POLB P06746 1/20 0.31
GPR139 Q6DWJ6 2/20 0.31
DRD2 P14416 1/20 0.31
ADRA1A P35348 1/20 0.31
DRD3 P35462 1/20 0.31
LMNA P02545 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
CENPE Q02224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8667760 0.99 MAPT (0.34) MAPTTHRBKMT2ABDKRB2POLB
Hydrochloric Acid SCHEMBL8670170 0.90 MAPT (0.34) MAPTTHRBKMT2ABDKRB2GPR139
SCHEMBL8669110 0.82 BDKRB2 (0.35) BDKRB2
SCHEMBL8475069 0.79 SMN1; SMN2 (0.37) MAPTTHRBKMT2APOLBGPR139
Hydrochloric Acid SCHEMBL8477672 0.78 SMN1; SMN2 (0.36) MAPTTHRBKMT2APOLBGPR139
SCHEMBL8671788 0.76 BDKRB2 (0.33) BDKRB2
SCHEMBL8667208 0.70 CENPE (0.35) BDKRB2CENPE
Hydrochloric Acid SCHEMBL8669829 0.69 CENPE (0.34) BDKRB2CENPE
SCHEMBL8669822 0.69 BDKRB2 (0.34) BDKRB2
SCHEMBL8559050 0.69 NPC1 (0.36) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750699-A HALOGENATING OF CORRESPONDING COMPOUND FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-05-12 US disclosed