SCHEMBL8669622

SCHEMBL8669622

CC(Nc1c(Nc2ccc3ncccc3c2)c(=O)c1=O)C(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 20/20 0.61
CHEK1 O14757 4/20 0.57
PLK4 O00444 3/20 0.57
DAPK3 O43293 3/20 0.57
ROCK2 O75116 3/20 0.57
CHEK2 O96017 3/20 0.57
PIM1 P11309 3/20 0.57
GSK3A P49840 3/20 0.57
ROCK1 Q13464 3/20 0.57
CDC42BPA Q5VT25 3/20 0.57
PLK3 Q9H4B4 3/20 0.57
CDC7 O00311 2/20 0.57
GSK3B P49841 2/20 0.57
PRKX P51817 2/20 0.57
CSNK1G2 P78368 2/20 0.57
PRKCZ Q05513 2/20 0.57
PKN2 Q16513 2/20 0.57
CLK4 Q9HAZ1 2/20 0.57
MKNK2 Q9HBH9 2/20 0.57
CSNK1G1 Q9HCP0 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357470 0.84 PLK1 (0.61) PLK1CHEK1PLK4DAPK3ROCK2
SCHEMBL7354053 0.83 PLK1 (0.50) PLK1CHEK1PLK4ROCK2CHEK2
SCHEMBL8674402 0.81 NPC1 (0.52) PLK1AURKASLK
SCHEMBL29120686 0.80 ALDH1A1 (0.59) SLK
SCHEMBL8672647 0.79 PLK1 (0.59) PLK1CHEK1PLK4DAPK3ROCK2
SCHEMBL29120687 0.78 ALDH1A1 (0.53) PLK1CHEK1PLK4DAPK3ROCK2
SCHEMBL29120695 0.77 NPC1 (0.61) ROCK2GSK3AROCK1GSK3BCLK4
SCHEMBL1927766 0.76 PLK1 (1.00) PLK1CHEK1PLK4DAPK3ROCK2
SCHEMBL1927178 0.76 PLK1 (1.00) PLK1CHEK1PLK4DAPK3ROCK2
SCHEMBL8668406 0.76 NPC1 (0.52) DYRK1ASLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729457-B1 DIAMINOCYCLOBUTENE-3,4-DIONES AS SMOOTH MUSCLE RELAXANTS AMERICAN HOME PROD (US) 1998-12-23 EP claimed