SCHEMBL8674402

SCHEMBL8674402

CNc1c(Nc2ccc3ncccc3c2)c(=O)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.52
POLB P06746 3/20 0.52
MAPT P10636 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
BRAF P15056 1/20 0.49
HTT P42858 3/20 0.48
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
ALDH1A1 P00352 4/20 0.47
RAB9A P51151 4/20 0.47
GRM4 Q14833 1/20 0.47
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PABPC1 P11940 1/20 0.47
PLK1 P53350 1/20 0.47
STK10 O94804 1/20 0.46
SLK Q9H2G2 1/20 0.46
EGFR P00533 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29120686 0.87 ALDH1A1 (0.59) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29120687 0.85 ALDH1A1 (0.53) NPC1POLBMAPTMEN1KMT2A
SCHEMBL7354053 0.85 PLK1 (0.50) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29120695 0.84 NPC1 (0.61) NPC1POLBMAPTMEN1KMT2A
SCHEMBL8668406 0.83 NPC1 (0.52) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29120691 0.82 IGF1R (0.54) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29120689 0.82 BRAF (0.47) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29120693 0.81 SYK (0.54) NPC1POLBMAPTMEN1KMT2A
SCHEMBL8669622 0.81 PLK1 (0.61) PLK1SLKAURKA
SCHEMBL3155590 0.80 NPC1 (0.62) NPC1POLBMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729457-B1 DIAMINOCYCLOBUTENE-3,4-DIONES AS SMOOTH MUSCLE RELAXANTS AMERICAN HOME PROD (US) 1998-12-23 EP claimed