SCHEMBL8670702

SCHEMBL8670702

CC(=O)Nc1ccc(Br)c2c1CC(N1CCCC1)CC2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
SLC18A3 Q16572 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
L3MBTL3 Q96JM7 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
CYP1A2 P05177 1/20 0.36
TP53 P04637 2/20 0.35
KDM2B Q8NHM5 1/20 0.35
HTR1D P28221 2/20 0.35
MBTD1 Q05BQ5 1/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8672548 0.79 SLC18A3 (0.52) NPC1SLC18A3HTR1DHTR1AHTR7
SCHEMBL30567319 0.75 RXFP1 (0.51) NPC1RXFP1TP53CA1CA2
SCHEMBL6674584 0.75 RXFP1 (0.51) NPC1RXFP1TP53CA1CA2
SCHEMBL2952459 0.75 RXFP1 (0.51) NPC1RXFP1TP53CA1CA2
SCHEMBL8668624 0.75 RXFP1 (0.40) NPC1SLC18A3RXFP1CYP1A2CA1
SCHEMBL8673705 0.74 MAPT (0.39) NPC1L3MBTL3L3MBTL1
SCHEMBL4199477 0.73 CYP1A2 (0.54) CYP1A2HTR1D
SCHEMBL4970280 0.73 CYP1A2 (0.54) CYP1A2HTR1D
SCHEMBL6785452 0.71 RXFP1 (0.44) NPC1RXFP1CA1CA2CA9
SCHEMBL7983593 0.70 RXFP1 (0.43) RXFP1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721234-A TREATING CONVULSIONS, ANXIETY, CEREBRAL HYPOXIA/ISCHEMIA, PARKINSON*S DISEASE WARNER-LAMBERT COMPANY (US) 1998-02-24 US disclosed
WO-1996017832-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYLQUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1996-06-13 WO disclosed