SCHEMBL8670723

SCHEMBL8670723

N#CCCC[CH]CCCCC#N

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 1/20 0.36
HIF1A Q16665 4/20 0.33
EPAS1 Q99814 4/20 0.33
LOX P28300 1/20 0.32
LOXL3 P58215 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6470309 0.94 TSHR (0.45) TSHRALDH1A1TDP1MAPTLOX
SCHEMBL11071480 0.92 ALDH1A1 (0.43) TSHRALDH1A1TDP1MAPTHIF1A
SCHEMBL29154624 0.88 ALDH1A1 (0.46) TSHRALDH1A1TDP1MAPTLOX
SCHEMBL14110162 0.83 TSHR (0.56) TSHRCYP3A4
SCHEMBL10486650 0.81
SCHEMBL8011581 0.80
SCHEMBL8723146 0.80
SCHEMBL59340 0.77
SCHEMBL30678315 0.77
SCHEMBL6000672 0.77 ALDH1A1 (0.64) TSHRALDH1A1TDP1MAPTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811422-A USEFUL FOR TREATING VIRAL INFECTIONS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-09-22 US disclosed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US disclosed
EP-0686151-A1 SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-12-13 EP disclosed