SCHEMBL8670902

SCHEMBL8670902

CCOC(=O)CCCCc1ccc(C#Cc2cc3c(cc2C)SCCC3(CC)CC)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4Z1 Q86W10 2/20 0.39
FFAR1 O14842 9/20 0.37
CYP3A4 P08684 1/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP4F11 Q9HBI6 1/20 0.36
CYP4F12 Q9HCS2 1/20 0.36
CHRM2 P08172 1/20 0.34
S1PR1 P21453 1/20 0.34
FPR1 P21462 1/20 0.34
FPR3 P25089 1/20 0.34
GPR183 P32249 1/20 0.34
APLNR P35414 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
GPR65 Q8IYL9 1/20 0.34
CYP4F2 P78329 2/20 0.33
CYP4A11 Q02928 2/20 0.33
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8659941 0.94 FFAR1 (0.41) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL8662589 0.93 CYP4Z1 (0.39) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL8674175 0.89 CYP3A4 (0.46) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL8674063 0.88 FDFT1 (0.40) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL7655279 0.88 CYP3A4 (0.42) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL7654882 0.86 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL8668889 0.85 CYP4F2 (0.36) CYP4Z1FFAR1CYP3A4RARARARB
SCHEMBL7648967 0.85 CYP4Z1 (0.32) CYP4Z1CYP3A4RARARARBRARG
SCHEMBL7651231 0.84 CYP4F2 (0.32) CYP4Z1CYP3A4RARARARBRARG
SCHEMBL7654485 0.84 CYP3A4 (0.37) CYP4Z1CYP3A4RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed