SCHEMBL8675665

SCHEMBL8675665

CCc1ccccc1N=C=O.O=C=Nc1cccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.46
GABRB2 P47870 3/20 0.46
CYP3A4 P08684 3/20 0.41
TRPA1 O75762 1/20 0.41
SIGMAR1 Q99720 5/20 0.34
TDP1 Q9NUW8 2/20 0.33
MAPK1 P28482 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8589377 0.92 GABRA1 (0.40) GABRA1GABRB2CYP3A4TRPA1SIGMAR1
SCHEMBL8943320 0.82 CYP3A4 (0.42) CYP3A4TRPA1TDP1MAPK1MEN1
SCHEMBL29795971 0.81 GABRA1 (0.61) GABRA1GABRB2CYP3A4TRPA1SIGMAR1
SCHEMBL93290 0.81 GABRA1 (0.61) GABRA1GABRB2CYP3A4TRPA1SIGMAR1
SCHEMBL59005 0.81 MAPK1 (0.45) GABRA1GABRB2CYP3A4TRPA1TDP1
SCHEMBL13645354 0.75 GABRA1 (0.44) GABRA1GABRB2CYP3A4TRPA1TDP1
SCHEMBL3843325 0.75 GABRA1 (0.44) GABRA1GABRB2CYP3A4TRPA1TDP1
SCHEMBL7757579 0.75 CYP3A4 (0.41) GABRA1GABRB2CYP3A4TRPA1SIGMAR1
SCHEMBL671741 0.74 CYP3A4 (0.54) GABRA1GABRB2CYP3A4TRPA1TDP1
SCHEMBL7001694 0.73 GABRA1 (0.52) GABRA1GABRB2CYP3A4TRPA1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880558-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-02 EP disclosed
WO-1997026300-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1997-07-24 WO disclosed