SCHEMBL8678902

SCHEMBL8678902

NC(=O)N1CCNCC1S(=O)(=O)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.50
CA2 P00918 6/20 0.50
CA9 Q16790 6/20 0.50
CA4 P22748 5/20 0.50
KMT2A Q03164 1/20 0.47
DPP4 P27487 3/20 0.39
CA5A P35218 1/20 0.38
DPP7 Q9UHL4 2/20 0.38
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 3/20 0.37
SLC6A2 P23975 2/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
F2 P00734 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061741 0.81 KMT2A (0.45) CA1CA2CA9CA4KMT2A
SCHEMBL3958698 0.80 CA1 (0.45) CA1CA2CA9CA4KMT2A
SCHEMBL20236395 0.78 CA1 (0.35) CA1CA2CA9CA4DPP4
SCHEMBL4584365 0.76 CA1 (0.63) CA1CA2CA9CA4DPP4
SCHEMBL6616045 0.75 KMT2A (0.43) CA1CA2CA9CA4KMT2A
SCHEMBL7357359 0.75 KMT2A (0.43) CA1CA2CA9CA4KMT2A
SCHEMBL3958464 0.71 CA1 (0.34) CA1CA2CA9CA4KMT2A
SCHEMBL2386164 0.71 DPP4 (0.47) CA1CA2CA9CA4DPP4
Hydrochloric Acid SCHEMBL28773228 0.70 DPP4 (0.46) CA1CA2CA9CA4KMT2A
SCHEMBL6744243 0.69 CA1 (0.44) CA1CA2CA9CA4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880512-A1 NOVEL AROMATIC PIPERAZINES DERIVED FROM SUBSTITUTED CYCLOAZANES, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITIONS, AND USE THEREOF AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1998-12-02 EP disclosed
WO-1997028141-A1 NOVEL AROMATIC PIPERAZINES DERIVED FROM SUBSTITUTED CYCLOAZANES, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITIONS, AND USE THEREOF AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed