SCHEMBL3958464

SCHEMBL3958464

CS(=O)(=O)C1CNCCN1C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA4 P22748 4/20 0.34
CA9 Q16790 4/20 0.34
APLNR P35414 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660031 0.84 CA1 (0.33) CA1CA2CA4CA9
SCHEMBL20236395 0.83 CA1 (0.35) CA1CA2CA4CA9
SCHEMBL3253967 0.83 CA1 (0.32) CA1CA2CA4CA9
SCHEMBL28071026 0.80 KDM4E (0.40) KDM4ECYP2D6
Hydrochloric Acid SCHEMBL5489333 0.79 CHRNB2 (0.37) CA1CA2CA4CA9KMT2A
SCHEMBL34472707 0.76 TP53 (0.32)
SCHEMBL954795 0.74 DPP4 (0.42) CA1CA2CA4CA9KDM4E
SCHEMBL954895 0.74 DPP4 (0.42) CA1CA2CA4CA9KDM4E
SCHEMBL11361171 0.74 APLNR (0.31) APLNR
SCHEMBL3958698 0.74 CA1 (0.45) CA1CA2CA4CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079756-A2 SYNTHETIC PEPTIDE AMIDES AND DIMERS THEREOF Cara Therapeutics, Inc. (US) 2009-07-22 EP disclosed
WO-2008060552-A2 SYNTHETIC PEPTIDE AMIDES AND DIMERS THEREOF CARA THERAPEUTICS, INC. (US) 2008-05-22 WO disclosed