SCHEMBL8679606

SCHEMBL8679606

C=C(C(=O)OC(=O)C(=C)c1ccc(OC(C)=O)c(OC(C)=O)c1)c1ccc(OC(C)=O)c(OC(C)=O)c1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.62
RAB9A P51151 2/20 0.62
KDM4E B2RXH2 1/20 0.62
ALDH1A1 P00352 1/20 0.62
GAA P10253 1/20 0.62
TOP1 P11387 3/20 0.51
PKM P14618 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NR3C1 P04150 1/20 0.42
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
CFD P00746 1/20 0.40
PTGS1 P23219 1/20 0.40
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TNFSF11 O14788 1/20 0.39
GAPDH P04406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8679604 0.88 TSHR (0.53) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL10767069 0.86 TSHR (0.66) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL6550416 0.78 TSHR (0.75) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL2219667 0.78 TSHR (0.64) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL3628967 0.78 TSHR (0.71) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL30154503 0.77 TSHR (1.00) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL640263 0.77 TSHR (1.00) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL2219672 0.77 GAA (0.62) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL8830836 0.75 TSHR (0.70) TSHRRAB9AKDM4EALDH1A1GAA
SCHEMBL10697221 0.75 TSHR (0.70) TSHRRAB9AKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712268-A Compositions of tricyclic β-lactams and uses thereof HOFFMANN-LA ROCHE INC. (US) 1998-01-27 US disclosed
US-5698577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1997-12-16 US disclosed
US-5510343-A BETA-LACTAMASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-04-23 US disclosed