SCHEMBL8681237

SCHEMBL8681237

Br[C]1C=Cc2ccccc2C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
TRPA1 O75762 3/20 0.38
CYP11B2 P19099 2/20 0.35
CYP11B1 P15538 1/20 0.35
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
MAOA P21397 3/20 0.33
MAOB P27338 2/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
PTGS2 P35354 1/20 0.32
TSHR P16473 1/20 0.31
HDAC3 O15379 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL283346 0.82 TRPA1 (0.50) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL31586332 0.82 TRPA1 (0.50) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL27986120 0.75 PARP1 (0.41) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL563921 0.74 TRPA1 (0.57) PARP1CA1CA2TRPA1BCHE
SCHEMBL11165595 0.73 CYP11B1 (0.37) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL23581856 0.71 PARP1 (0.39) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL10546236 0.71 PARP1 (0.39) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL3900328 0.71 PARP1 (0.39) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL23581853 0.71 PARP1 (0.39) PARP1CA1CA2TRPA1CYP11B2
SCHEMBL10546234 0.71 CA1 (0.42) PARP1CA1CA2TRPA1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843983-A Diphenylethane compounds containing a saturated heterocyclic group, their preparation, and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1998-12-01 US disclosed
CN-1174190-A Diaryl alkane derivatives containing alicyclic group, their preparation and their therapeutic and prophylactic uses SANKYO CO (JP) 1998-02-25 CN disclosed
EP-0790235-A1 Diaryl alkane derivatives containing an alicyclic group, their preparation and their therapeutic and prophylactic uses SANKYO COMPANY LIMITED (JP) 1997-08-20 EP disclosed