SCHEMBL8682014

SCHEMBL8682014

OC(c1nccs1)(c1nccs1)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.52
NR1H2 P55055 1/20 0.47
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 3/20 0.37
PRKDC P78527 1/20 0.37
ALDH1A1 P00352 4/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
HIF1A Q16665 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TSHR P16473 1/20 0.36
NOS1 P29475 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.35
FBP1 P09467 2/20 0.33
PDK1 Q15118 1/20 0.33
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8682291 0.83 AR (0.46) ARNR1H2MEN1KMT2AMAPT
SCHEMBL16230730 0.83 AR (0.43) ARNR1H2ALDH1A1TSHRNOS1
SCHEMBL5759768 0.83 AR (0.42) ARNR1H2MEN1KMT2AMAPT
SCHEMBL8617994 0.82 AR (0.53) ARNR1H2MEN1KMT2AMAPT
SCHEMBL26229838 0.79 AR (0.40) ARNR1H2MEN1KMT2AMAPT
SCHEMBL6288482 0.79 AR (0.42) ARNR1H2MEN1KMT2AMAPT
SCHEMBL8617770 0.79 AR (0.50) ARNR1H2PRKDCFBP1ALOX5
SCHEMBL27837232 0.78
SCHEMBL9434229 0.78 AR (0.55) ARNR1H2PRKDCALOX5
SCHEMBL31478751 0.77 ALDH1A1 (0.39) ARNR1H2MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843971-A 1, 1-BIS (heteroazolyl) alkane derivatives and their use as neuroprotective agents ASTRA AKTIEBOLAG (SE) 1998-12-01 US claimed
WO-1995033747-A1 NOVEL 1,1-BIS(HETEROAZOLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS ASTRA AKTIEBOLAG (SE) 1995-12-14 WO claimed
US-5843971-A 1, 1-BIS (heteroazolyl) alkane derivatives and their use as neuroprotective agents ASTRA AKTIEBOLAG (SE) 1998-12-01 US disclosed
US-5665747-A TREATING NERVOUS SYSTEM, PSYCHOLOGICAL, AND BRAIN DISORDERS ASTRA AKTIEBOLAG (SE) 1997-09-09 US disclosed
EP-0765325-A1 NOVEL 1,1-BIS(HETEROAZOLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS Astra Aktiebolag (SE) 1997-04-02 EP disclosed
WO-1995033747-A1 NOVEL 1,1-BIS(HETEROAZOLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS ASTRA AKTIEBOLAG (SE) 1995-12-14 WO disclosed