SCHEMBL8683290

SCHEMBL8683290

O=c1ncc(-c2ccc(Cl)cc2)c[nH]1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.52
MAP4K4 O95819 2/20 0.48
MCL1 Q07820 1/20 0.44
NOTUM Q6P988 2/20 0.43
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
EIF4E P06730 1/20 0.41
AKT2 P31751 6/20 0.41
GAA P10253 3/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
TSHR P16473 1/20 0.40
METAP2 P50579 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
RUNX1 Q01196 1/20 0.40
CBFB Q13951 1/20 0.40
CCNT1 O60563 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12863970 0.81 LYN (0.44) HSD11B1NOTUMKDM4EALDH1A1GAA
SCHEMBL12864123 0.80 NOTUM (0.41) HSD11B1NOTUMEIF4EAKT2AKT1
SCHEMBL2352218 0.80 AKT1 (0.52) MAP4K4MCL1NOTUMKDM4EALDH1A1
SCHEMBL10898482 0.79 IDO1 (0.50) MAP4K4NOTUMKDM4E
SCHEMBL7223891 0.78 MYLK4 (0.37) HSD11B1KDM4EEIF4E
SCHEMBL9822966 0.78 EIF4E (0.45) HSD11B1MAP4K4KDM4EEIF4E
SCHEMBL10898602 0.77 ALDH1A1 (0.50) KDM4EALDH1A1MAPTTHRBCCNT1
SCHEMBL7232041 0.77 AXL (0.49) MAP4K4KDM4EALDH1A1EIF4E
SCHEMBL5070333 0.75 MAPT (0.56) MCL1NOTUMKDM4EALDH1A1GAA
SCHEMBL8616381 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753642-A AGRICULTURE, MEDICINE ROHM AND HAAS COMPANY (US) 1998-05-19 US disclosed
US-5728698-A AGRICULTURAL USE, RICE, WHEAT ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728694-A Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728715-A FOR MAMMALS, AGRICULTURE, RICE, WHEAT, TOMATOES ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5726162-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5726176-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5631254-A RICE; HUMAN INFECTIONS ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
US-5552409-A PHYTOPATHOGENIC, RICE ROHM AND HAAS COMPANY (US) 1996-09-03 US disclosed
EP-0478195-A1 Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1992-04-01 EP disclosed
US-4613603-A Compounds with a nitrogen-containing heterocyclic nucleus, and drugs in which they are present SANOFI (FR) 1986-09-23 US disclosed