SCHEMBL8684841

SCHEMBL8684841

CCC(=O)C(=C(SC)SC)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.57
CES2 O00748 5/20 0.57
RAB9A P51151 3/20 0.46
LMNA P02545 3/20 0.46
MAPT P10636 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 2/20 0.46
XBP1 P17861 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
HPGD P15428 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
ATM Q13315 1/20 0.39
TP53 P04637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2376839 0.80 MAPT (0.58) CES1CES2RAB9ALMNAMAPT
SCHEMBL12985768 0.78 CES1 (0.59) CES1CES2RAB9ALMNAMAPT
SCHEMBL7669290 0.73 CES2 (1.00) CES1CES2RAB9ALMNAMAPT
SCHEMBL4625390 0.73 CES2 (1.00) CES1CES2RAB9ALMNAMAPT
SCHEMBL6206988 0.72 CES1 (0.55) CES1CES2RAB9ALMNAMAPT
SCHEMBL9818176 0.69 CES1 (0.52) CES1CES2RAB9ALMNAMAPT
SCHEMBL9710316 0.69 CES1 (0.63) CES1CES2RAB9ALMNAMAPT
SCHEMBL31175926 0.69 CES2 (0.76) CES1CES2RAB9ALMNAMAPT
SCHEMBL27908851 0.69 CES1 (0.52) CES1CES2RAB9ALMNAMAPT
SCHEMBL5698372 0.69 CES1 (0.52) CES1CES2RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750560-A ANTICOAGULANTS; FREE RADICAL SCAVENGERS; CARDIOVASCULAR, GASTROINTESTINAL, NERVOUS SYSTEM AND RESPIRATORY SYSTEM DISORDERS LABORATOIRES DE THERAPEUTIQUE MODERNE (FR) 1998-05-12 US disclosed
US-5470871-A Free radical scavengers, microbiocides and calcium or potassium channel activators for cardiovascular disorders, nervous system disorders or respiratory system disorders LABORATOIRES DE THERAPEUTIQUE MODERNE (FR) 1995-11-28 US disclosed