SCHEMBL8687366

SCHEMBL8687366

CC(=NOCCOC1SC(=O)N(Cc2ccccc2)C1=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.44
MAPT P10636 7/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
PPARG P37231 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 4/20 0.40
HPGD P15428 1/20 0.40
THRB P10828 3/20 0.39
GAA P10253 1/20 0.39
PPARA Q07869 2/20 0.39
TP53 P04637 1/20 0.38
EP300 Q09472 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689520 0.81 POLB (0.35) POLBMAPTL3MBTL1PPARGMAPK1
SCHEMBL8686882 0.78 ALDH1A1 (0.37) POLBMAPTPPARGHTTALDH1A1
SCHEMBL3774754 0.77 MAPT (0.50) POLBMAPTALDH1A1THRBGAA
SCHEMBL6032173 0.76 MAPT (0.54) POLBMAPTL3MBTL1ALDH1A1THRB
SCHEMBL8689646 0.74 POLB (0.40) POLBMAPTL3MBTL1PPARGLMNA
SCHEMBL8687292 0.74 TAAR1 (0.41) POLBMAPTLMNAMAPK1HTT
SCHEMBL7469304 0.73 POLB (0.55) POLBMAPTL3MBTL1ALDH1A1THRB
SCHEMBL8689551 0.73 POLB (0.41) POLBMAPTL3MBTL1LMNAMAPK1
SCHEMBL8523889 0.73 POLB (0.47) POLBMAPTL3MBTL1ALDH1A1HPGD
SCHEMBL8687360 0.72 PPARG (0.48) MAPTL3MBTL1PPARGLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780490-A A O-(2,4-OXA(OR THIA)ZOLIDINYL)PHENYLOXY(OR THIO OR AMINO) ALKYLOXIME; ALDOSE REDUCTASE INHIBITORS; ANTIDIABETIC AND -HYPOGLYCEMIC AGENTS; LIVER, SKIN AND UROGENITAL DISORDERS SANKYO COMPANY, LIMITED (JP) 1998-07-14 US disclosed
US-5703096-A ANTIDIABETIC AGENTS; ALDOSE REDUCTASE INHIBITOR SANKYO COMPANY, LIMITED (JP) 1997-12-30 US disclosed