SCHEMBL8687733

SCHEMBL8687733

CCCN(C)c1ccc(-c2cnc[nH]2)c2c1OCO2

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 10/20 0.38
ADRA2B P18089 3/20 0.37
ADRA2C P18825 3/20 0.37
ADRA1A P35348 3/20 0.37
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
IDO1 P14902 6/20 0.33
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8687765 0.75 CYP1A2 (0.37) HSP90AA1HSP90AB1CYP1A2CYP3A4CYP2D6
SCHEMBL8687758 0.69 IDO1 (0.39) ADRA2AADRA2BADRA2CADRA1ACYP1A2
SCHEMBL8687342 0.68 CYP1A2 (0.40) CYP1A2CYP3A4CYP2D6IDO1
SCHEMBL26259980 0.57 IDO1 (0.64) ADRA2AADRA2BCYP3A4CYP2D6IDO1
SCHEMBL7194641 0.54 IDO1 (0.59) CYP3A4CYP2D6IDO1
SCHEMBL10707409 0.54 MEN1 (0.35)
SCHEMBL27490016 0.54 IDO1 (0.67) ADRA2ACYP3A4IDO1
SCHEMBL16921858 0.54 HCAR3 (0.35)
SCHEMBL1950240 0.53 IDO1 (0.64) HSP90AA1HSP90AB1CYP1A2CYP3A4CYP2D6
SCHEMBL16997427 0.53 ALDH1A1 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807860-A ACYLCOENZYME A:CHOLESTEROL ACYLTRANSFERASE INHIBITORS; HYPERLIPEMIA, ATHEROSCLEROSIS; ANTICHOLESTEROL AGENTS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-09-15 US disclosed
EP-0773218-A1 N-(Piperazinylalkoxyphenyl)-N'phenylalkylurea derivatives as ACAT inhibitors for the treatment of atheroschlerosis MITSUBISHI CHEMICAL CORPORATION (JP) 1997-05-14 EP disclosed