SCHEMBL8688339

SCHEMBL8688339

Oc1ccc(-c2nccn2Cc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK2 P53671 1/20 0.59
HSD17B10 Q99714 2/20 0.55
BRD4 O60885 2/20 0.53
ESR1 P03372 1/20 0.50
ALDH1A1 P00352 3/20 0.49
KMT2A Q03164 3/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
HSP90AA1 P07900 1/20 0.48
PDE6D O43924 1/20 0.46
PLAA Q9Y263 1/20 0.45
ALPG P10696 1/20 0.44
FDPS P14324 1/20 0.44
MEN1 O00255 2/20 0.43
HTR6 P50406 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX12 P18054 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5981532 0.89 LIMK2 (0.63) LIMK2HSD17B10BRD4ESR1ALDH1A1
SCHEMBL17621 0.89 HSD17B10 (0.62) LIMK2HSD17B10BRD4ESR1ALDH1A1
Iodide SCHEMBL28519464 0.87 HSD17B10 (0.60) LIMK2HSD17B10BRD4ESR1ALDH1A1
Hydrochloric Acid SCHEMBL233781 0.87 HSD17B10 (0.60) LIMK2HSD17B10BRD4ESR1ALDH1A1
Fluoride SCHEMBL10339918 0.87 HSD17B10 (0.60) LIMK2HSD17B10BRD4ESR1ALDH1A1
Bromide SCHEMBL811908 0.87 HSD17B10 (0.60) LIMK2HSD17B10BRD4ESR1ALDH1A1
Fluoride Ion SCHEMBL10906965 0.85 LIMK2 (0.59) LIMK2HSD17B10BRD4ESR1ALDH1A1
Fluoride SCHEMBL10906966 0.85 LIMK2 (0.59) LIMK2HSD17B10BRD4ESR1ALDH1A1
Bromide SCHEMBL811907 0.85 LIMK2 (0.59) LIMK2HSD17B10BRD4ESR1ALDH1A1
SCHEMBL3155427 0.84 LIMK2 (0.59) LIMK2HSD17B10BRD4ESR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719169-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
EP-0640593-B1 Substituted benzoylguanidines, process for their preparation, their use as medicine or in diagnostic and medicines containing them HOECHST AG (DE) 1997-12-29 EP disclosed
EP-0640593-A1 Substituted benzoylguanidines, process for their preparation, their use as medicine or in diagnostic and medicines containing them HOECHST AKTIENGESELLSCHAFT (DE) 1995-03-01 EP disclosed