SCHEMBL8689248

SCHEMBL8689248

COc1ccc(-c2cc(CO)nn2-c2ccccc2S(N)(=O)=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 14/20 0.67
CA1 P00915 13/20 0.67
CA2 P00918 13/20 0.67
PTGS2 P35354 6/20 0.51
CHRNA7 P36544 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5798707 0.88 CA9 (0.65) CA9CA1CA2PTGS2
SCHEMBL6406740 0.87 CA9 (0.66) CA9CA1CA2PTGS2
SCHEMBL8677688 0.85 CA1 (0.52) CA9CA1CA2PTGS2
SCHEMBL8015867 0.85 PTGS2 (0.65) CA9CA1CA2PTGS2
SCHEMBL6307500 0.85 CA1 (0.49) CA9CA1CA2PTGS2CHRNA7
SCHEMBL8730045 0.85 CA9 (0.49) CA9CA1CA2PTGS2
SCHEMBL8688670 0.84 CA1 (0.48) CA9CA1CA2PTGS2
SCHEMBL8420267 0.84 PTGS2 (0.58) CA9CA1CA2PTGS2
SCHEMBL8689144 0.81 PTGS2 (0.48) CA9CA1CA2PTGS2CHRNA7
SCHEMBL28301021 0.81 CA1 (0.55) CA9CA1CA2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed