SCHEMBL8690601

SCHEMBL8690601

COc1ccc(C(C)(O)c2ocnc2C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.38
AHR P35869 2/20 0.37
ALDH1A1 P00352 3/20 0.36
PKM P14618 1/20 0.36
MAPT P10636 2/20 0.36
HSD11B1 P28845 1/20 0.35
CYP19A1 P11511 1/20 0.35
LMNA P02545 2/20 0.35
ALOX15 P16050 1/20 0.35
APEX1 P27695 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27344981 0.83 ALDH1A1 (0.46) ALDH1A1PKMMAPTLMNAMAPK1
SCHEMBL9260610 0.82 ALDH1A1 (0.36) AOC3ALDH1A1PKMMAPTLMNA
SCHEMBL8688642 0.81 CYP3A4 (0.41) ALDH1A1MAPTLMNAALOX15MAPK1
Fluoride Ion SCHEMBL8981546 0.79 ALDH1A1 (0.34) AOC3ALDH1A1PKMMAPTLMNA
SCHEMBL8981551 0.77 ALDH1A1 (0.33) AOC3AHRALDH1A1PKMMAPT
SCHEMBL7128923 0.74 CA1 (0.55) AOC3ALDH1A1MAPTHSD11B1LMNA
SCHEMBL28076770 0.71 ACHE (0.62) AOC3ALDH1A1MAPTHSD11B1LMNA
SCHEMBL25485515 0.71 ACHE (0.62) AOC3ALDH1A1MAPTHSD11B1LMNA
SCHEMBL29226506 0.70 AOC3 (0.41) AOC3AHRALDH1A1MAPTHSD11B1
SCHEMBL30927963 0.70 AOC3 (0.41) AOC3AHRALDH1A1MAPTHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747515-A Heterocyclic compounds and compositions having nevropharmacological potential ASTRA AKTIEBOLAG (SE) 1998-05-05 US claimed
US-5747515-A Heterocyclic compounds and compositions having nevropharmacological potential ASTRA AKTIEBOLAG (SE) 1998-05-05 US disclosed
EP-0707573-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001967-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed