SCHEMBL8691306

SCHEMBL8691306

Nc1c(F)ccc2nc(Cl)sc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
CDK5 Q00535 2/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CDK5R1 Q15078 1/20 0.35
DYRK1A Q13627 2/20 0.34
AURKA O14965 1/20 0.34
DAPK3 O43293 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
NTRK1 P04629 1/20 0.34
PDGFRA P16234 1/20 0.34
PRKACA P17612 1/20 0.34
LTK P29376 1/20 0.34
GRK5 P34947 1/20 0.34
MAPK8 P45983 1/20 0.34
CSNK1A1 P48729 1/20 0.34
CDK8 P49336 1/20 0.34
CLK2 P49760 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20969710 0.81 ACACB (0.36) ALDH1A1CDK5CCNE1CDK2CDK5R1
SCHEMBL8693683 0.81 SMN1; SMN2 (0.41) ALDH1A1MAPTCDK5DYRK1AAURKA
SCHEMBL27370484 0.78 MAPT (0.43) ALDH1A1MAPTCDK5DYRK1AAURKA
SCHEMBL8688516 0.78 SMN1; SMN2 (0.44) ALDH1A1MAPTCCNE1CDK2AXL
SCHEMBL19709636 0.78 ALDH1A1 (0.33) ALDH1A1CDK5CCNE1CDK2CDK5R1
SCHEMBL27379338 0.77 ALDH1A1 (0.38) ALDH1A1MAPTCDK5CCNE1CDK2
SCHEMBL20969721 0.73 KDM4E (0.42) ALDH1A1MAPTCDK5DYRK1AAURKA
SCHEMBL20969585 0.73 ACACB (0.36) ALDH1A1MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL4242805 0.73 PSMB8 (0.43) ALDH1A1MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL8689714 0.71 ARNT (0.38) ALDH1A1MAPTCDK5CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753595-A Herbicidal 3-(substituted benzoxazol-7-yl) and 3-(Substituted benzothiazol-7-yl)-1-substituted-6-trifluoromethyl-2 4-(1h 3h)pyrimidinediones FMC CORPORATION (US) 1998-05-19 US disclosed
WO-1997008170-A1 HERBICIDAL 3-(SUBSTITUTED BENZOXAZOL-7-YL) AND 3-(SUBSTITUTED BENZOTHIAZOL-7-YL)-1-SUBSTITUTED-6-TRIFLUOROMETHYL-2,4-(1H,3H)PYRIMIDINEDIONES FMC CORPORATION (US) 1997-03-06 WO disclosed