SCHEMBL8693757

SCHEMBL8693757

O=c1c2ncccc2c(-c2ccc3c(c2)OCO3)nn1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.51
ALDH1A1 P00352 7/20 0.48
GAA P10253 1/20 0.47
PDE4A P27815 4/20 0.47
PDE4B Q07343 4/20 0.47
PDE4C Q08493 4/20 0.47
PDE4D Q08499 4/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK1 P28482 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
EDNRB P24530 1/20 0.45
EDNRA P25101 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365746 0.93 PDE4A (0.56) PDE5AALDH1A1GAAPDE4APDE4B
SCHEMBL7359586 0.92 PDE4A (0.57) PDE5AALDH1A1GAAPDE4APDE4B
SCHEMBL7364301 0.86 HTT (0.47) PDE5AALDH1A1GAAPDE4ACYP1A2
SCHEMBL7361880 0.85 PDE4A (0.67) PDE5AALDH1A1GAAPDE4APDE4B
SCHEMBL7369761 0.82 ALDH1A1 (0.70) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7368929 0.82 TSHR (0.50) ALDH1A1GAAPDE4APDE4BPDE4C
SCHEMBL7364759 0.82 PDE4A (0.52) PDE5AALDH1A1GAAPDE4APDE4B
SCHEMBL7363442 0.80 PDE4A (0.71) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7366591 0.79 ALDH1A1 (0.59) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL7369583 0.79 ALDH1A1 (0.56) ALDH1A1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed