SCHEMBL8694071

SCHEMBL8694071

CCN(CC)C(=O)c1ccccc1[S+]([O-])C1=C(C(=O)O)N2C(=O)[C@H](C(C)O)[C@@H]2[C@H]1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
PTGS1 P23219 1/20 0.40
PDE4A P27815 1/20 0.40
ABCC2 Q92887 1/20 0.39
KEAP1 Q14145 1/20 0.34
CACNA1C Q13936 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
ELANE P08246 1/20 0.31
HPGD P15428 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
MAPT P10636 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8039652 1.00 ESR1 (0.40) ESR1PTGS1PDE4AABCC2KEAP1
SCHEMBL8695696 1.00 ESR1 (0.40) ESR1PTGS1PDE4AABCC2KEAP1
SCHEMBL8699086 0.88 ESR1 (0.31) ESR1PTGS1PDE4AABCC2KEAP1
SCHEMBL8975950 0.86 ESR1 (0.42) ESR1PTGS1PDE4AABCC2CACNA1C
SCHEMBL8040731 0.85 ELANE (0.32) ELANE
SCHEMBL8046000 0.82 ELANE (0.38) ELANERAB9ASMN1; SMN2
SCHEMBL8576696 0.80 PTGS1 (0.42) ESR1PTGS1PDE4AABCC2CACNA1C
SCHEMBL9836778 0.80 PTGS1 (0.42) ESR1PTGS1PDE4AABCC2CACNA1C
SCHEMBL9128902 0.80 PTGS1 (0.42) ESR1PTGS1PDE4AABCC2CACNA1C
SCHEMBL8700514 0.78 ESR1 (0.42) ESR1PTGS1PDE4AABCC2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719275-A REACTING SILYL ENOL ETHER WITH AZETIDINONE DERIVATIVE TO FORM INTERMEDIATE FOR PENICILLIN-TYPE ANTIBIOTIC SANKYO COMPANY, LIMITED (JP) 1998-02-17 US disclosed