SCHEMBL8695907

SCHEMBL8695907

NC(N)(Cc1ccccc1)C(=O)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.57
HIF1A Q16665 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CES2 O00748 1/20 0.50
AKR1B1 P15121 1/20 0.50
SLC6A2 P23975 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
PTPN1 P18031 1/20 0.46
PAM P19021 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
FNTA P49354 1/20 0.42
FNTB P49356 1/20 0.42
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42
SLC7A5 Q01650 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29787058 0.84 ALDH1A1 (0.49) CES1HIF1ASMN1; SMN2SLC6A2PTPN1
SCHEMBL1081531 0.81 SMN1; SMN2 (0.69) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL5647919 0.81 SLC6A2 (0.53) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL12902954 0.78 CES1 (0.59) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL3761802 0.76 SMN1; SMN2 (0.57) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL16816903 0.75 SMN1; SMN2 (0.67) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL2336417 0.75 SMN1; SMN2 (0.67) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL17498702 0.75 SMN1; SMN2 (0.67) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL29187272 0.74 CES1 (0.55) CES1HIF1ASMN1; SMN2CES2AKR1B1
SCHEMBL215167 0.73 CES1 (0.53) CES1HIF1ASMN1; SMN2CES2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760248-A HAVING IMPROVED METABOLIC STABILITY A.MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-06-02 US disclosed
WO-1995015311-A1 TACHYKININ ANTAGONISTS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1995-06-08 WO disclosed