SCHEMBL8697199

SCHEMBL8697199

CCOC(=O)Oc1[nH]c2c3ccccc3n(C)c2c1-c1ccc(OC)cc1OCCO.CCOC(=O)Oc1c(-c2ccc(OC)cc2OCCO)c2c(c3ccccc3n2C)n1Cc1ccc2nsnc2c1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 5/20 0.39
EDNRA P25101 2/20 0.33
PTPN1 P18031 2/20 0.32
PPARG P37231 2/20 0.31
TP53 P04637 2/20 0.30
RXFP1 Q9HBX9 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8698594 0.85 PTPN1 (0.39) EDNRBPTPN1TP53
SCHEMBL8697633 0.78 POLB (0.37) EDNRBPTPN1
SCHEMBL8697275 0.78 PTPN1 (0.42) EDNRBPTPN1
SCHEMBL8697591 0.77 PTPN1 (0.46) PTPN1TP53
SCHEMBL8697402 0.74 NTRK1 (0.39)
SCHEMBL8702544 0.73 EDNRB (0.38) EDNRBPTPN1TP53
SCHEMBL8547930 0.73 EDNRB (0.47) EDNRBEDNRAPTPN1PPARG
SCHEMBL8704430 0.72 EDNRB (0.34) EDNRBPTPN1
SCHEMBL8551472 0.72 EDNRB (0.43) EDNRBEDNRAPTPN1TP53
SCHEMBL8549234 0.72 EDNRB (0.52) EDNRBEDNRAPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042709-A1 ENDOTHELIN-RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-10-01 WO disclosed