SCHEMBL8697214

SCHEMBL8697214

O=C(c1ccc(F)cc1)c1ccc2[nH]c(=S)oc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 7/20 0.59
KEAP1 Q14145 1/20 0.47
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPK1 P28482 2/20 0.41
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
GAA P10253 1/20 0.41
CREBBP Q92793 1/20 0.40
LTA4H P09960 1/20 0.40
SMYD3 Q9H7B4 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
PTGS1 P23219 1/20 0.39
KDR P35968 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697822 0.87 PSMB8 (0.63) PSMB8KEAP1KDM4EALDH1A1MEN1
SCHEMBL8697342 0.85 PSMB8 (0.64) PSMB8KEAP1KDM4EALDH1A1KMT2A
SCHEMBL8697415 0.85 PSMB8 (0.64) PSMB8KEAP1KDM4EALDH1A1KMT2A
SCHEMBL118689 0.80 PSMB8 (0.68) PSMB8KEAP1KDM4EALDH1A1MEN1
SCHEMBL8698103 0.79 PSMB8 (0.59) PSMB8KEAP1KDM4EALDH1A1GAA
SCHEMBL16150847 0.79 PSMB8 (0.61) PSMB8KEAP1KDM4EALDH1A1MEN1
SCHEMBL8701858 0.75 PSMB8 (0.54) PSMB8KEAP1KDM4EALDH1A1KMT2A
SCHEMBL1094167 0.75 PSMB8 (0.65) PSMB8KEAP1KDM4EALDH1A1MEN1
SCHEMBL8704890 0.74 PSMB8 (0.53) PSMB8KEAP1KDM4EALDH1A1KMT2A
SCHEMBL8698800 0.73 PSMB8 (0.52) PSMB8KEAP1KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025913-A1 NOVEL SUBSTITUTED 3H -BENZOXAZOLE-2-THIONES AND 3H -BENZOTHIAZOLE-2 THIONES DERIVATIVES, METHOD FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1998-06-18 WO disclosed