SCHEMBL8698563

SCHEMBL8698563

Cn1c(=S)oc2cc(C(O)c3ccccn3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
MAPT P10636 4/20 0.37
CYP3A4 P08684 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
CYP2C9 P11712 2/20 0.37
ALDH1A1 P00352 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CYP2C19 P33261 1/20 0.36
KMO O15229 3/20 0.35
KAT7 O95251 1/20 0.35
KAT6A Q92794 1/20 0.35
RECQL P46063 1/20 0.35
MIF P14174 1/20 0.34
PKM P14618 1/20 0.34
SLC6A3 Q01959 2/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
LMNA P02545 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703947 0.82 MIF (0.41) ALDH1A1KDM4EMIFPKMHTT
SCHEMBL8704872 0.76 ALDH1A1 (0.42) BRD4MAPTALDH1A1KDM4EMIF
SCHEMBL8701154 0.72 PSMB8 (0.43) BRD4MAPTTDP1ALDH1A1KDM4E
SCHEMBL14081505 0.66 BRD4 (0.49) BRD4MAPTCYP3A4CYP2C9ALDH1A1
SCHEMBL29485027 0.66 BRD4 (0.49) BRD4MAPTCYP3A4CYP2C9ALDH1A1
SCHEMBL23610040 0.66 BRD4 (0.49) BRD4MAPTCYP3A4CYP2C9ALDH1A1
SCHEMBL1602617 0.66 SLC6A2 (0.40) BRD4MAPTCYP3A4ALDH1A1KMO
SCHEMBL9003879 0.66 BRD4 (0.46) BRD4MAPTCYP3A4ALDH1A1KDM4E
SCHEMBL31143703 0.66 BRD4 (0.46) BRD4MAPTCYP3A4ALDH1A1KDM4E
SCHEMBL30392540 0.66 BRD4 (0.46) BRD4MAPTCYP3A4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025913-A1 NOVEL SUBSTITUTED 3H -BENZOXAZOLE-2-THIONES AND 3H -BENZOTHIAZOLE-2 THIONES DERIVATIVES, METHOD FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1998-06-18 WO disclosed