SCHEMBL8698709

SCHEMBL8698709

CCCCn1cc(C(=O)OCC)c(NC(=S)Nc2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
GAA P10253 4/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
RAB9A P51151 3/20 0.53
NPC1 O15118 3/20 0.53
MAPT P10636 6/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
ALOX12 P18054 3/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HPGD P15428 3/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KDM4E B2RXH2 2/20 0.44
F2 P00734 1/20 0.44
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693075 0.89 NPC1 (0.47) ALDH1A1SMN1; SMN2GAAL3MBTL1RAB9A
SCHEMBL8693750 0.84 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2GAARAB9ANPC1
SCHEMBL8699774 0.84 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2GAARAB9ANPC1
SCHEMBL8694579 0.84 KMT2A (0.39) ALDH1A1SMN1; SMN2GAAL3MBTL1RAB9A
SCHEMBL8698386 0.82 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2GAARAB9ANPC1
SCHEMBL8696818 0.81 HTT (0.41) ALDH1A1RAB9ANPC1MEN1KMT2A
SCHEMBL8694568 0.80 TEAD2 (0.39) ALDH1A1SMN1; SMN2GAAL3MBTL1MAPT
SCHEMBL8693986 0.80 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2GAARAB9ANPC1
SCHEMBL8692506 0.80 TEAD2 (0.39) ALDH1A1SMN1; SMN2GAAL3MBTL1MAPT
SCHEMBL8693117 0.79 MAPT (0.50) ALDH1A1GAARAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed