SCHEMBL8133151

SCHEMBL8133151

CCCN(CCC)C1CCc2cc(NC(C)=O)c(Br)cc2C1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.57
DRD3 P35462 9/20 0.51
DRD2 P14416 7/20 0.51
DRD4 P21917 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
HTR1A P08908 2/20 0.51
ADRB2 P07550 1/20 0.51
CYP2D6 P10635 1/20 0.51
CASP1 P29466 1/20 0.51
LMNA P02545 2/20 0.50
MAPT P10636 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7494029 0.85 FYN (0.51) FYNDRD3DRD2DRD4MEN1
SCHEMBL7494035 0.85 FYN (0.51) FYNDRD3DRD2DRD4MEN1
SCHEMBL8124799 0.79 DRD2 (0.56) DRD3DRD2DRD4HTR1AADRB2
SCHEMBL9776784 0.79 DRD2 (0.63) FYNDRD3DRD2DRD4MEN1
SCHEMBL7503050 0.79 DRD3 (0.60) FYNDRD3DRD2DRD4MEN1
Bromide SCHEMBL10975000 0.78 DRD2 (0.64) FYNDRD3DRD2DRD4MEN1
SCHEMBL8128394 0.76 FYN (0.63) FYNDRD3DRD2DRD4MEN1
SCHEMBL7330393 0.75 DRD2 (0.64) DRD3DRD2DRD4HTR1AADRB2
SCHEMBL9759545 0.75 HTR1A (0.64) DRD3DRD2HTR1ACYP2D6LMNA
SCHEMBL8699267 0.75 CA1 (0.38) MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690843-B1 Formyl- or cyano- substituted indole derivatives having dopaminergic activity UPJOHN CO (US) 2000-08-30 EP disclosed