SCHEMBL8699456

SCHEMBL8699456

CC(C)(C)OC(=O)NCN1CCC[C@H]1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
ACE P12821 1/20 0.42
EPHX1 P07099 1/20 0.42
HSD17B10 Q99714 2/20 0.41
BTK Q06187 1/20 0.40
LMNA P02545 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KLK5 Q9Y337 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20545129 0.86 EPHX1 (0.46) SMN1; SMN2ACEEPHX1HSD17B10BTK
SCHEMBL3266228 0.83 EPHX1 (0.43) SMN1; SMN2EPHX1KMT2AMEN1ALDH1A1
SCHEMBL27483297 0.81 ALDH1A1 (0.37) SMN1; SMN2ACEEPHX1HSD17B10LMNA
SCHEMBL29283308 0.81 EPHX1 (0.41) SMN1; SMN2ACEEPHX1HSD17B10KMT2A
SCHEMBL16279605 0.78 TDP1 (0.48) EPHX1KMT2AMEN1CA1CA2
SCHEMBL16279606 0.78 TDP1 (0.48) EPHX1KMT2AMEN1CA1CA2
SCHEMBL1925210 0.78 ACE (0.53) SMN1; SMN2ACEHSD17B10BTKLMNA
SCHEMBL1000948 0.78 ACE (0.53) SMN1; SMN2ACEHSD17B10BTKLMNA
SCHEMBL19022219 0.78 HSD17B10 (0.47) SMN1; SMN2ACEHSD17B10LMNACYP2C19
SCHEMBL1912615 0.78 HSD17B10 (0.47) SMN1; SMN2ACEHSD17B10LMNACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5741799-A ANTICOAGULANTS OF SULFONAMIDO HETEROCYCLIC THROMBIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-04-21 US disclosed
US-5741792-A ANTICOAGULANTS OF SULFONAMIDO HETEROCYCLIC THROMBIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-04-21 US disclosed
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0623596-A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-09 EP disclosed