SCHEMBL8699549

SCHEMBL8699549

Cc1ccc(S(=O)(=O)O)cc1.N[C@@H]1C=CC[C@@H]2CN(c3ncc4c(=O)c(C(=O)O)cn(C5CC5)c4c3Cl)C[C@@H]21

nearest known ligand 0.40

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 1/20 0.40
ALDH1A1 P00352 3/20 0.40
POLB P06746 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRD1 P41143 1/20 0.40
DPP4 P27487 5/20 0.36
KCNH2 Q12809 5/20 0.34
TOP2A P11388 3/20 0.33
TOP2B Q02880 3/20 0.33
KDM4E B2RXH2 2/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
HPGD P15428 1/20 0.32
XBP1 P17861 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693108 0.91 ALDH1A1 (0.42) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7851593 0.91 ALDH1A1 (0.31) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7852422 0.90 POLB (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL8695363 0.89 ALDH1A1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
Bromide SCHEMBL8693293 0.89 ALDH1A1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8695572 0.89 ALDH1A1 (0.41) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7851071 0.84 ALDH1A1 (0.37) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8693112 0.83 ALDH1A1 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7841322 0.82 ALDH1A1 (0.33) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7851419 0.81 ALDH1A1 (0.41) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811433-A ANTIMICROBIALS BAYER AKTIENGESELLSCHAFT (DE) 1998-09-22 US disclosed