SCHEMBL8700129

SCHEMBL8700129

CC1=C(C(=O)O)C(c2ccccc2F)C(C(=O)O)=C(C)N1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.54
NR1I2 O75469 1/20 0.45
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 5/20 0.43
CACNA1B Q00975 4/20 0.43
HSD17B10 Q99714 4/20 0.43
HPGD P15428 3/20 0.43
TP53 P04637 3/20 0.43
KMT2A Q03164 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
ABCC4 O15439 1/20 0.43
PLIN1 O60240 1/20 0.43
CACNA1F O60840 1/20 0.43
GMNN O75496 1/20 0.43
KCNK2 O95069 1/20 0.43
ABCB11 O95342 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953639 0.87 GAA (0.45) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL27673576 0.85 MAPT (0.56) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL6950016 0.84 ALOX15 (0.50) ALDH1A1KDM4ECACNA1BCACNA1FADORA3
SCHEMBL27544295 0.83 TSHR (0.46) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL8222248 0.83 GAA (0.43) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL2615091 0.83 NR1I2 (0.65) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL29676427 0.83 NR1I2 (0.65) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL2615090 0.83 NR1I2 (0.65) GAANR1I2ALDH1A1KDM4ECACNA1B
SCHEMBL9235674 0.82 CACNA1B (0.46) CACNA1BCACNA1FADORA3CACNA1DCACNA1S
SCHEMBL3027183 0.80 ADORA3 (0.59) GAANR1I2ALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7196614-A None JP disclosed
CN-114516774-A Preparation method of chiral bromo-1, 4-dihydropyridine compound 中国科学院成都生物研究所 2022-05-20 CN disclosed
CN-1089337-C 1, 4-dihydropyridine derivatives MERCIAN CORP (JP) 2002-08-21 CN disclosed
US-5760238-A ANTIISCHEMIC AGENTS MERCIAN CORPORATION (JP) 1998-06-02 US disclosed
CN-1156450-A 1,4-dihydropyridine derivatives MERCIAN CORP (JP) 1997-08-06 CN disclosed
JP-H07196614-A PHENYL-SUBSTITUTED 1,4-DIHYDROPYRIDINE BAYER AG 1995-08-01 JP disclosed
US-4699984-A Preparation of intermediates to 6-fluoro-7-(2,6-dimethylpyridyl)quinoline carboxylic acids and compounds STERLING DRUG INC. (US) 1987-10-13 US disclosed
EP-0179239-A2 7-(Pyridinyl)-/-alkyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid having antibacterial activity and preparation thereof STERLING DRUG INC. (US) 1986-04-30 EP disclosed