SCHEMBL8700142

SCHEMBL8700142

Cc1c(C(=O)N=C(N)N)ccc(-c2cccnc2)c1S(C)(=O)=O

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
PTGS2 P35354 1/20 0.42
SLC9A1 P19634 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27376941 0.86 PTGS2 (0.44) MKNK1MKNK2PTGS2
SCHEMBL8446139 0.85 PTGS2 (0.40) MKNK1MKNK2PTGS2SLC9A1
SCHEMBL8528490 0.81 SLC9A1 (0.53) SLC9A1
SCHEMBL8180285 0.80 SLC9A1 (0.38) SLC9A1
SCHEMBL8702013 0.80 SLC2A1 (0.49) MKNK1MKNK2PTGS2
SCHEMBL8699934 0.79 SLC9A1 (0.40) SLC9A1
SCHEMBL8532248 0.78 SLC9A1 (0.48) SLC9A1
SCHEMBL8444418 0.76 SLC9A1 (0.54) SLC9A1
SCHEMBL8446483 0.76 SLC9A1 (0.54) SLC9A1
SCHEMBL8533825 0.76 SLC9A1 (0.55) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753680-A Heterocyclyl-benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-19 US disclosed
EP-0699666-A1 Heterocyclic substituted benzoylguanidine MERCK PATENT GmbH (DE) 1996-03-06 EP disclosed