SCHEMBL8700368

SCHEMBL8700368

CC(=O)CCc1nc2[nH]c(=O)[nH]c(=O)c2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
ADORA2B P29275 1/20 0.40
XDH P47989 3/20 0.38
ENPP1 P22413 1/20 0.36
ACHE P22303 1/20 0.35
GDA Q9Y2T3 1/20 0.35
RECQL P46063 1/20 0.34
PARP1 P09874 2/20 0.34
PARP2 Q9UGN5 2/20 0.34
POLB P06746 2/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
P2RY12 Q9H244 2/20 0.33
BLM P54132 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9721482 0.89 CYP2C19 (0.41) MAPTADORA2BXDHENPP1POLB
SCHEMBL7326384 0.85 MAPT (0.43) MAPTADORA2BXDHENPP1ACHE
SCHEMBL7530553 0.81 MAPT (0.46) MAPTADORA2BXDHENPP1ACHE
SCHEMBL1150739 0.81 XDH (0.47) MAPTADORA2BXDHACHEGDA
SCHEMBL6233162 0.79 XDH (0.51) MAPTADORA2BXDHPARP1ALDH1A1
SCHEMBL31438586 0.78 MAPT (0.48) MAPTADORA2BXDHENPP1ACHE
SCHEMBL380136 0.78 MAPT (0.48) MAPTADORA2BXDHACHEGDA
SCHEMBL3118423 0.77 XDH (0.54) MAPTADORA2BXDHPARP1
SCHEMBL541696 0.77 MAPT (0.42) MAPTADORA2BXDHACHEGDA
SCHEMBL11661802 0.76 XDH (0.56) MAPTXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710272-A INCREASING CEREBRAL BLOOD FLOW HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5472873-A Rhodotorula rubra useful in a process for the preparation of (ω-1)-hydroxyalkylxanthines HOECHST AKTIENGESELLSCHAFT (DE) 1995-12-05 US disclosed
US-5310666-A Vascular disorders HOECHST AKTIENGESELLSCHAFT (DE) 1994-05-10 US disclosed