SCHEMBL8700563

SCHEMBL8700563

Cn1c(=O)oc2cc(C(=O)c3ccccc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 1.00
HPGD P15428 1/20 1.00
SIGMAR1 Q99720 1/20 0.65
SMN1; SMN2 Q16637 2/20 0.60
GLA P06280 1/20 0.60
ASAH1 Q13510 2/20 0.52
POLB P06746 3/20 0.51
TP53 P04637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PKM P14618 3/20 0.50
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 1/20 0.48
KDM4E B2RXH2 1/20 0.48
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565098 0.88 ALDH1A1 (0.79) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL14565048 0.87 ALDH1A1 (0.77) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL9683762 0.86 ALDH1A1 (0.76) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL14565012 0.86 ALDH1A1 (0.75) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
Hydrochloric Acid SCHEMBL9683732 0.85 ALDH1A1 (0.73) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL474056 0.84 ALDH1A1 (0.73) ALDH1A1HPGDSIGMAR1SMN1; SMN2POLB
SCHEMBL8703282 0.84 ALDH1A1 (0.72) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL9616042 0.84 ALDH1A1 (0.72) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL14565009 0.83 ALDH1A1 (0.71) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA
SCHEMBL14565011 0.83 ALDH1A1 (0.70) ALDH1A1HPGDSIGMAR1SMN1; SMN2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070054899-A1 Aromatase inhibitor compounds and uses thereof PARALLEL WIRELESS, INC. 2007-03-08 US disclosed
US-20070054899-A1 Aromatase inhibitor compounds and uses thereof PARALLEL WIRELESS, INC. 2007-03-08 US disclosed
WO-1998025913-A1 NOVEL SUBSTITUTED 3H -BENZOXAZOLE-2-THIONES AND 3H -BENZOTHIAZOLE-2 THIONES DERIVATIVES, METHOD FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1998-06-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054899-A1 Aromatase inhibitor compounds and uses thereof CYP19A1, CYP17A1, HSD17B11 ALDH1A1 207/4885HPGD 155/4885SIGMAR1 3852/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.