SCHEMBL8700930

SCHEMBL8700930

CCCCC(=O)N(C)c1c(N)ccn(-c2ccc(-c3ccccc3-c3nnn[nH]3)cc2)c1=O

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 5/20 0.37
AGTR1 P30556 12/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ABCB11 O95342 1/20 0.34
GP6 Q9HCN6 1/20 0.34
AGTR2 P50052 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8260354 0.73 LTB4R2 (0.52) LTB4R2AGTR1ABCB11GP6
SCHEMBL8092930 0.73 LTB4R2 (0.49) LTB4R2AGTR1ABCB11GP6
SCHEMBL9486277 0.73 LTB4R2 (0.44) LTB4R2AGTR1AGTR2
SCHEMBL2976631 0.71 AGTR1 (0.53) LTB4R2AGTR1ABCB11GP6AGTR2
SCHEMBL684200 0.70 LTB4R2 (0.50) LTB4R2AGTR1ABCB11GP6
SCHEMBL28463355 0.70 LTB4R2 (0.51) LTB4R2AGTR1ABCB11GP6
SCHEMBL2969136 0.70 AGTR1 (0.58) LTB4R2AGTR1ABCB11GP6AGTR2
SCHEMBL2969141 0.70 AGTR1 (0.54) LTB4R2AGTR1ABCB11GP6AGTR2
SCHEMBL18425480 0.69 LTB4R2 (0.69) LTB4R2AGTR1
SCHEMBL14051316 0.69 AGTR1 (0.44) LTB4R2AGTR1ABCB11GP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5798364-A ANGIOTENSIN II ANTAGONIST, USEFUL FOR TREATMENT OF HYPERTENSION, ALDOSTERONISM AND CARDIAC INSUFFICIENCY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-08-25 US disclosed