SCHEMBL8701925

SCHEMBL8701925

Fc1ccc(C(c2cc3ccccc3o2)n2cnnc2)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.52
CYP26A1 O43174 2/20 0.39
CYP17A1 P05093 1/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 2/20 0.36
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP24A1 Q07973 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697624 0.84 CYP19A1 (0.50) CYP19A1CYP26A1CYP17A1TSHR
SCHEMBL8698220 0.83 CYP19A1 (0.69) CYP19A1CYP26A1NPC1TSHRMAPK1
SCHEMBL8697755 0.81 CYP19A1 (0.73) CYP19A1CYP26A1CYP3A4
SCHEMBL8696281 0.76 CYP19A1 (0.56) CYP19A1CYP26A1NPC1RAB9ACYP24A1
SCHEMBL8702874 0.76 IDO1 (0.35) CYP19A1NPC1RAB9AMEN1KMT2A
SCHEMBL8697952 0.76 IDO1 (0.33) NPC1RAB9ATSHRCYP3A4MEN1
SCHEMBL8697855 0.75 CYP19A1 (0.40) CYP19A1NPC1RAB9ATSHRMAPK1
SCHEMBL8700053 0.73 CYP19A1 (0.51) CYP19A1CYP26A1CYP17A1TSHR
SCHEMBL8696295 0.72 CYP19A1 (0.65) CYP19A1CYP26A1NPC1RAB9A
SCHEMBL8696639 0.72 CYP19A1 (0.73) CYP19A1CYP26A1CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed