SCHEMBL8702178

SCHEMBL8702178

O=C=Nc1cc(C(F)(F)F)cs1.O=C=Nc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.34
SERPINE1 P05121 2/20 0.32
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
NOS3 P29474 2/20 0.31
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
EPHX2 P34913 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591338 0.83 TRPA1 (0.37) CYP3A4
SCHEMBL3974623 0.82
SCHEMBL180952 0.80 TSHR (0.45) TRPV1CYP3A4TSHRNOS3NOS1
SCHEMBL7728817 0.77 TRPA1 (0.32) CYP3A4
SCHEMBL7357034 0.76 KIF11 (0.45) SERPINE1CYP3A4TSHRNOS3NOS1
SCHEMBL10968174 0.71
SCHEMBL24246067 0.70 MAPK1 (0.41) CYP3A4TSHRNOS3NOS1NOS2
SCHEMBL10546748 0.70 CYP3A4 (0.41) CYP3A4TSHREPHX2
SCHEMBL10967071 0.70
SCHEMBL9859153 0.69 CYP3A4 (0.44) CYP3A4TSHRNOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998008813-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED PYRROLIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed