SCHEMBL8709376

SCHEMBL8709376

COc1ccc(NC(C)=S)c(C)c1C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.42
HPGD P15428 3/20 0.42
EPHX1 P07099 1/20 0.42
TSHR P16473 2/20 0.41
HTT P42858 2/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 2/20 0.39
KMT2A Q03164 4/20 0.38
MAPT P10636 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
MEN1 O00255 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2C P18825 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5409015 0.81 ALDH1A1 (0.59) ALDH1A1HPGDEPHX1TSHRHTT
SCHEMBL12702785 0.74 APP (0.42) ALDH1A1TSHRGAAKMT2AMAPT
SCHEMBL30601570 0.73 HPGD (0.66) ALDH1A1HPGDHTTGAAKDM4E
SCHEMBL3129401 0.73 HPGD (0.66) ALDH1A1HPGDHTTGAAKDM4E
SCHEMBL24356362 0.73 ALDH1A1 (0.77) ALDH1A1HPGDGAAKMT2AMAPT
SCHEMBL29793327 0.72 ACHE (0.52) ALDH1A1HPGDTSHRGAAKDM4E
SCHEMBL1635785 0.72 ACHE (0.52) ALDH1A1HPGDTSHRGAAKDM4E
SCHEMBL25210284 0.71 ALDH1A1 (0.51) ALDH1A1HPGDEPHX1HTTGAA
SCHEMBL4778825 0.69 PDE4B (0.43) ALDH1A1HPGDTSHRGAAKDM4E
SCHEMBL10886977 0.69 ALDH1A1 (0.51) ALDH1A1HPGDHTTGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1252717-A Intermediate and method for preparing benzo [ b ] thiophene LILLY CO ELI (US) 2000-05-10 CN disclosed
WO-1998048787-A1 INTERMEDIATES AND A PROCESS FOR PREPARING BENZO[b]THIOPHENES ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed