SCHEMBL8709443

SCHEMBL8709443

N#Cc1cccc(N)c1.N#Cc1cccc(N2CCNCC2)c1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.85
DRD3 P35462 2/20 0.85
ADRB1 P08588 4/20 0.51
HTR1A P08908 3/20 0.51
HTR7 P34969 3/20 0.51
HTR3E A5X5Y0 3/20 0.51
HTR3B O95264 3/20 0.51
HTR3A P46098 3/20 0.51
HTR3D Q70Z44 3/20 0.51
HTR3C Q8WXA8 3/20 0.51
SIGMAR1 Q99720 3/20 0.51
HTR2C P28335 3/20 0.51
THRB P10828 2/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A4 P31645 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30855584 0.92 DRD2 (1.00) DRD2DRD3ADRB1HTR1AHTR7
SCHEMBL249732 0.92 DRD2 (1.00) DRD2DRD3ADRB1HTR1AHTR7
Hydrochloric Acid SCHEMBL6408589 0.91 DRD2 (0.97) DRD2DRD3ADRB1HTR1AHTR7
Hydrochloric Acid SCHEMBL29882147 0.91 DRD2 (0.97) DRD2DRD3ADRB1HTR1AHTR7
Hydrochloric Acid SCHEMBL6494513 0.91 DRD2 (0.97) DRD2DRD3ADRB1HTR1AHTR7
SCHEMBL20159295 0.86 DRD2 (0.88) DRD2DRD3ADRB1HTR1AHTR7
Hydrochloric Acid SCHEMBL20141804 0.85 DRD2 (0.85) DRD2DRD3ADRB1HTR1AHTR7
SCHEMBL29922419 0.84 HTR7 (0.65) DRD2DRD3ADRB1HTR1AHTR7
Piperazine SCHEMBL27880049 0.84 DRD2 (0.56) DRD2DRD3CYP3A4SLC6A4
SCHEMBL112735 0.84 HTR7 (0.65) DRD2DRD3ADRB1HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002432-A1 BICYCLIC COMPOUNDS FOR CONTROLLING MICTURITION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-22 WO disclosed