SCHEMBL8710070

SCHEMBL8710070

NC(=O)OCCCO[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA4 P22748 5/20 0.46
CA9 Q16790 5/20 0.46
PTGS2 P35354 1/20 0.40
LMNA P02545 2/20 0.39
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
CHRM5 P08912 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
HTR1A P08908 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
CHRNA7 P36544 1/20 0.38
GLA P06280 1/20 0.36
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712167 0.87 LMNA (0.40) CA12CA1CA2CA4CA9
SCHEMBL16914733 0.83 CA12 (0.45) CA12CA1CA2CA4CA9
SCHEMBL16914736 0.81 CA12 (0.44) CA12CA1CA2CA4CA9
SCHEMBL23036023 0.79 CA12 (0.43) CA12CA1CA2CA4CA9
SCHEMBL21105278 0.79 ALDH1A1 (0.50) CA12CA1CA2CA4CA9
SCHEMBL23036025 0.79 CA12 (0.43) CA12CA1CA2CA4CA9
SCHEMBL2745809 0.79 LMNA (0.52) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL4731008 0.79 CA12 (0.48) CA12CA1CA2CA4CA9
SCHEMBL13018462 0.79 CHRM2 (0.34) CA12CA1CA2CA4CA9
SCHEMBL2014045 0.78 CA12 (0.41) CA12CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed