SCHEMBL871014

SCHEMBL871014

CCOC(=O)c1cn2cc(C)ccc2n1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.69
POLB P06746 1/20 0.69
RAB9A P51151 6/20 0.59
GAA P10253 2/20 0.58
ALDH1A1 P00352 2/20 0.54
HPGD P15428 2/20 0.54
NPC1 O15118 4/20 0.53
MAPT P10636 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
RXFP1 Q9HBX9 1/20 0.53
CYP1A2 P05177 1/20 0.53
GABRA2 P47869 2/20 0.52
GABRB2 P47870 2/20 0.52
KMT2A Q03164 2/20 0.52
GLA P06280 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118658 0.88 KDM4E (0.66) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL1500236 0.86 KDM4E (0.64) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL4098270 0.86 KDM4E (0.64) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL70705 0.86 KDM4E (0.64) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL3545619 0.86 KDM4E (0.64) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL741904 0.86 KDM4E (0.64) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL21246447 0.85 RAB9A (0.52) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL21033471 0.85 KDM4E (0.63) KDM4EPOLBRAB9AGAAALDH1A1
Hydrochloric Acid SCHEMBL21223028 0.85 KDM4E (0.63) KDM4EPOLBRAB9AGAAALDH1A1
SCHEMBL8608432 0.85 KDM4E (0.63) KDM4EPOLBRAB9AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119528903-A Compounds for the treatment of spinal muscular atrophy PTC医疗公司 2025-02-28 CN disclosed
CN-108299314-B Compounds for the treatment of spinal muscular atrophy PTC医疗公司 2024-11-26 CN disclosed
CN-118434744-A Nitrogen-containing macrocyclic compound, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-08-02 CN disclosed
WO-2024059186-A1 N-((ISOQUINOLIN-6-YL)METHYL)-1H-PYRAZOLE-4-CARBOXAMID DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS FOR THE TREATMENT OF HEREDITARY ANGIOEDEMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-03-21 WO disclosed
WO-2024046512-A2 NITROGEN-CONTAINING MACROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 中国医药研究开发中心有限公司 2024-03-07 WO disclosed
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. 2024-02-29 US disclosed
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. 2024-02-29 US disclosed
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. 2024-02-29 US disclosed
EP-4289838-A2 ARYLMETHOXY ISOINDOLINE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME Celgene Corporation (US) 2023-12-13 EP disclosed
US-11753407-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2023-09-12 US disclosed
US-20050171092-A1 Chemical compounds ASTRAZENECA AB, A SWEDEN CORPORATION 2005-08-04 US disclosed
EP-1274701-B1 [1,4']-BIPIPERIDINE COMPOUNDS ASTRAZENECA AB (SE) 2005-06-29 EP disclosed
US-6903115-B2 Bipiperidine compounds ASTRAZENECA AB (SE) 2005-06-07 US disclosed
EP-1493743-A1 Substituted bipiperidine intermediates and derivatives thereof AstraZeneca AB (SE) 2005-01-05 EP disclosed
US-20040014783-A1 Chemical compounds ASTRAZENECA AB, A SWEDEN CORPORATION 2004-01-22 US disclosed
US-20040006080-A1 Chemical compounds ASTRAZENECA AB, A SWEDEN CORPORATION 2004-01-08 US disclosed
US-6525070-B2 For therapy of chemokine (such as CCR3) or H1 mediated disease state ASTRAZENECA AB (SE) 2003-02-25 US disclosed
EP-1274701-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2003-01-15 EP disclosed
US-20020077337-A1 Chemical compounds ASTRAZENECA AB (SE) 2002-06-20 US disclosed
WO-2001077101-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2001-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 KDM4E 2384/4885POLB 1579/4885RAB9A 1350/4885
US-20020077337-A1 Chemical compounds CCR3, CCR1, CCR4 KDM4E 3900/4885POLB 3341/4885RAB9A 2344/4885
US-20050171092-A1 Chemical compounds CCR3, CCR1, CCR4 KDM4E 3589/4885POLB 3244/4885RAB9A 2189/4885
US-20040006080-A1 Chemical compounds CCR3, CCR1, CCR4 KDM4E 3900/4885POLB 3341/4885RAB9A 2344/4885
US-20040014783-A1 Chemical compounds CCR3, CCR1, CCR4 KDM4E 3900/4885POLB 3341/4885RAB9A 2344/4885
US-11753407-B2 Compounds for treating spinal muscular atrophy SMN1; SMN2, CPT1B, GYS1 KDM4E 1370/4885POLB 1594/4885RAB9A 1386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.