SCHEMBL8710945

SCHEMBL8710945

CC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)OCc1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.72
POLB P06746 1/20 0.55
TSHR P16473 1/20 0.54
MDM4 O15151 1/20 0.54
MDM2 Q00987 1/20 0.54
CTSS P25774 2/20 0.54
CTSK P43235 2/20 0.54
CTSL P07711 1/20 0.54
CTSB P07858 1/20 0.54
ACE P12821 1/20 0.53
PAM P19021 1/20 0.52
ALDH1A1 P00352 1/20 0.52
ALOX15 P16050 1/20 0.52
MBTPS1 Q14703 1/20 0.52
MAPT P10636 1/20 0.51
S1PR1 P21453 1/20 0.51
TYR P14679 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710942 1.00 TACR1 (0.72) TACR1POLBTSHRMDM4MDM2
SCHEMBL30621980 0.94 TACR1 (0.80) TACR1POLBCTSSCTSKCTSL
SCHEMBL5887474 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL5887859 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL2853641 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL2853645 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL5887863 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL5887473 0.89 TACR1 (0.69) TACR1POLBCTSSCTSKACE
SCHEMBL8765789 0.88 CTSL (0.58) TACR1POLBTSHRMDM4MDM2
SCHEMBL3065366 0.87 CTSL (0.64) TACR1CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116947858-A Compounds selectively inhibiting four amino acid modifications of ADP, preparation and application thereof 首都医科大学 2023-10-27 CN claimed
CN-116947858-A Compounds selectively inhibiting four amino acid modifications of ADP, preparation and application thereof 首都医科大学 2023-10-27 CN disclosed
US-5776902-A Boronophenyl analogs of phospholyrosines TRUSTEES OF TUFTS UNIVERSITY (US) 1998-07-07 US disclosed
WO-1995025118-A2 INHIBITORS OF SH2 DOMAIN INTERACTIONS TRUSTEES OF TUFTS UNIVERSITY (US) 1995-09-21 WO disclosed