SCHEMBL8710971

SCHEMBL8710971

Cc1ccc(NC(=O)c2ccc([N+](=O)[O-])cc2)cc1C

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.80
MAPT P10636 7/20 0.80
KMT2A Q03164 6/20 0.80
MEN1 O00255 5/20 0.80
NPC1 O15118 5/20 0.67
ALDH1A1 P00352 2/20 0.67
TDP1 Q9NUW8 2/20 0.61
MITF O75030 2/20 0.61
POLB P06746 2/20 0.61
HTT P42858 4/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
LMNA P02545 3/20 0.60
ATM Q13315 2/20 0.60
MAPK1 P28482 2/20 0.60
KDM4E B2RXH2 1/20 0.58
FKBP5 Q13451 1/20 0.57
HPGD P15428 1/20 0.56
CASP3 P42574 2/20 0.56
CASP2 P42575 1/20 0.56
CASP7 P55210 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16728064 0.88 KMT2A (0.74) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL29145506 0.87 MEN1 (0.74) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL29145514 0.86 RAB9A (0.72) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL23898948 0.84 KMT2A (0.83) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL9134339 0.84 KMT2A (0.83) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL8572381 0.84 KMT2A (0.83) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL12406969 0.83 KMT2A (0.71) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL20313717 0.83 KMT2A (0.71) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL8713449 0.83 KMT2A (0.71) RAB9AMAPTKMT2AMEN1NPC1
SCHEMBL1249138 0.82 KMT2A (0.63) RAB9AMAPTKMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed