SCHEMBL8712669

SCHEMBL8712669

CC(C)=CCOS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.50
MMP1 P03956 2/20 0.44
MMP9 P14780 2/20 0.44
MMP13 P45452 2/20 0.44
STAT3 P40763 2/20 0.43
TLR9 Q9NR96 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2D6 P10635 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
ALDH1A1 P00352 4/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
MMP2 P08253 1/20 0.39
MMP8 P22894 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622204 0.87 TRPV1 (0.58) DHODHTRPV1ALDH1A1
SCHEMBL3092862 0.87 TRPV1 (0.58) DHODHTRPV1ALDH1A1
SCHEMBL23802602 0.85 TRPV1 (0.56) DHODHKMT2AMAPK1TRPV1ALDH1A1
SCHEMBL8058501 0.85 TRPV1 (0.56) DHODHKMT2AMAPK1TRPV1ALDH1A1
SCHEMBL15246442 0.85 TRPV1 (0.56) DHODHKMT2AMAPK1TRPV1ALDH1A1
SCHEMBL8058497 0.85 TRPV1 (0.56) DHODHKMT2AMAPK1TRPV1ALDH1A1
SCHEMBL27733182 0.85 TRPV1 (0.56) DHODHKMT2AMAPK1TRPV1ALDH1A1
SCHEMBL30218691 0.84 POLB (0.42) DHODHKMT2ASMN1; SMN2LMNAMAPK1
SCHEMBL1018380 0.83 DHODH (0.40) DHODHMMP1MMP9MMP13STAT3
SCHEMBL1018381 0.83 DHODH (0.40) DHODHMMP1MMP9MMP13STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107298667-B Method for synthesizing icaritin 北京盛诺基医药科技股份有限公司 2020-09-08 CN claimed
CN-107216303-B Synthesis method of fluccoladine 北京盛诺基医药科技股份有限公司 2020-04-21 CN claimed
CN-107216302-B Synthesis method of flucloratadine 北京盛诺基医药科技股份有限公司 2020-02-21 CN claimed
CN-107216303-B Synthesis method of fluccoladine 北京盛诺基医药科技股份有限公司 2020-04-21 CN disclosed
EP-0613877-B1 Preparation process of quinone derivative and intermediate for the preparation thereof EISAI KAGAKU KK (JP) 1998-05-20 EP disclosed
US-5686635-A Tetrahydro-alkenyl-methanonaphthalene-5,8-dione derivatives EISAI CHEMICAL CO., LTD. (JP) 1997-11-11 US disclosed
US-5677471-A Process for the preparation of quinone derivative EISAI CHEMICAL CO., LTD. (JP) 1997-10-14 US disclosed
US-5476955-A Process for the preparation of a quinone derivative EISAI CHEMICAL CO., LTD. (JP) 1995-12-19 US disclosed
EP-0613877-A1 Preparation process of quinone derivative and intermediate for the preparation thereof EISAI CHEMICAL CO., LTD. (JP) 1994-09-07 EP disclosed