SCHEMBL8712694

SCHEMBL8712694

COC(CN(C)C(=O)c1ccc(C(=O)N2CCN(c3ncccc3NC(C)C)CC2)cc1)OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
MAOA P21397 1/20 0.45
TBXA2R P21731 1/20 0.45
OPRM1 P35372 1/20 0.45
MDH1 P40925 1/20 0.45
KCNH2 Q12809 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SLC6A7 Q99884 7/20 0.40
HSD11B1 P28845 1/20 0.40
GPR6 P46095 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7861562 0.90 ADRA2A (0.42) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8709684 0.86 ADRA2A (0.47) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8714403 0.86 ADRA2A (0.47) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8709879 0.85 ADRA2A (0.46) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8713960 0.83 ADRA2A (0.47) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8710321 0.83 ADRA2A (0.44) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8711077 0.83 OPRM1 (0.51) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8708456 0.83 NAMPT (0.47) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8711887 0.83 ADRA2A (0.51) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8709600 0.81 ADRA2A (0.54) ADRA2AADORA3CHRM1MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998054140-A1 NOVEL TEREPHTHALAMIDE DERIVATIVES DONGWHA PHARMACEUTICAL IND. CO., LTD. (KR) 1998-12-03 WO disclosed