SCHEMBL8713101

SCHEMBL8713101

N/N=C1\Nc2ccccc2C(c2ccccc2)=NC1NC(=O)CCC1CCCCC1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.59
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HDAC1 Q13547 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CCKBR P32239 10/20 0.45
CCKAR P32238 8/20 0.45
OXTR P30559 1/20 0.43
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8608811 1.00 KCNH2 (0.59) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL8608963 0.91 KCNH2 (0.60) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL7090389 0.91 KCNH2 (0.60) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL7090394 0.91 KCNH2 (0.60) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL8801265 0.88 KCNH2 (0.56) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL8801258 0.88 KCNH2 (0.56) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL7213180 0.86 KCNH2 (0.63) KCNH2ALDH1A1MEN1KMT2ATDP1
SCHEMBL17467746 0.75 CCKBR (0.54) CCKBRCCKAR
SCHEMBL7090700 0.74 KCNH2 (1.00) KCNH2HDAC1CCKBRCCKARPSEN1
SCHEMBL7087129 0.74 KCNH2 (1.00) KCNH2HDAC1CCKBRCCKARPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817658-A ADMINISTERING A DIAZEPINE COMPOUND; DISEASES OF THE EAR MERCK & COMPANY, INC. (US) 1998-10-06 US disclosed